Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetAdenosine receptor A3(Homo sapiens (Human))
Universitat Wurzburg

Curated by PDSP Ki Database
LigandPNGBDBM50041895(2-substituted NECA derivatives, 4 | 5-[6-Amino-2-(...)
Affinity DataKi:  4.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universitat Wurzburg

Curated by PDSP Ki Database
LigandPNGBDBM50041895(2-substituted NECA derivatives, 4 | 5-[6-Amino-2-(...)
Affinity DataKi:  14nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Universitat Wurzburg

Curated by PDSP Ki Database
LigandPNGBDBM50041895(2-substituted NECA derivatives, 4 | 5-[6-Amino-2-(...)
Affinity DataKi:  40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50453355(CHEMBL2113408)
Affinity DataKi:  70nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50453355(CHEMBL2113408)
Affinity DataEC50:  6.05E+3nMAssay Description:Negative chronotropic activity via A1 Adenosine receptor was tested in spontaneously beating rat atriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed