Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Pfizer

Curated by ChEMBL

LigandBDBM50349460(CHEMBL1808580)Copy SMILESCopy InChI

Affinity DataIC50:  2.14E+4nMAssay Description:Inhibition of TPL2 using GST-MEK as substrate by LANCE assayMore data for this Ligand-Target Pair

Target InfoPDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI