Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetKelch-like ECH-associated protein 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50130557(CHEMBL3632882)
Affinity DataIC50:  85nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) protein-protein interaction expressed in Escherichia coli BL21 codon plus cells using FITC-beta-DEETGEF-OH ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKelch-like ECH-associated protein 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50130557(CHEMBL3632882)
Affinity DataIC50:  400nMAssay Description:Binding affinity to the Keap1 (321 to 609 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by surface plasmon resonance assa...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKelch-like ECH-associated protein 1(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50130557(CHEMBL3632882)
Affinity DataKd:  400nMAssay Description:Inhibition of Keap1-Nrf2 (unknown origin) protein-protein interaction by SPR assayMore data for this Ligand-Target Pair
In DepthDetails PubMed