Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50205510((S,R)-(-)-ethyl {4-[2-{[2-(3-bromoisoxazol-5-yl)-2...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I]CYP from human adrenergic beta 2 receptor transfected in CHO cells in presence of 100 uM GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50205510((S,R)-(-)-ethyl {4-[2-{[2-(3-bromoisoxazol-5-yl)-2...)
Affinity DataKi:  23nMAssay Description:Displacement of [125I]CYP from human adrenergic beta 1 receptor transfected in CHO cells in presence of 100 uM GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50205510((S,R)-(-)-ethyl {4-[2-{[2-(3-bromoisoxazol-5-yl)-2...)
Affinity DataKi:  1.01E+4nMAssay Description:Displacement of [125I]CYP from human adrenergic beta 3 receptor transfected in CHO cells in presence of 100 uM GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed