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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50173987((9-Carbamoyl-4-{4-[2-(3,4-difluoro-phenyl)-ethyl]-...)
Affinity DataIC50:  122nMAssay Description:Inhibition of MRP1 in human COR-L23/R cells assessed reduction in tritiated daunomycin efflux incubated for 2 hrs by radioactivity-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50173987((9-Carbamoyl-4-{4-[2-(3,4-difluoro-phenyl)-ethyl]-...)
Affinity DataIC50: <250nMAssay Description:Inhibitory concentration against multidrug resistance associated protein 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed