Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 2 hits in this display
IC50: 3.50E+3nMAssay Description:Inhibition of human ERG assessed as decrease in tail current amplitude measured after 5 mins by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
EC50: 15nMAssay Description:Partial agonist activity at human M4 receptor co-expressed with Galpha16 in CHO cells assessed as calcium mobilization after 60 mins by FLIPR assayMore data for this Ligand-Target Pair