Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hit in this display   

TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Heptares Therapeutics

US Patent

LigandBDBM280406(US10030012, Example 36 | ethyl 4-[4-(2- methylpyri...)Copy SMILESCopy InChI

Affinity DataEC50:  6.73E+3nMAssay Description:The functional activity of compounds at the M4 and M2 receptors was determined by measuring changes in the level of intracellular calcium ions caused...More data for this Ligand-Target Pair

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