Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetAdenosine receptor A1(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50072943(CHEMBL3410310)
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cells by Top Count analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50072943(CHEMBL3410310)
Affinity DataKi:  4.30E+3nMAssay Description:Displacement of [3H]HEMADO from human adenosine A3 receptor expressed in CHO cells by Top Count analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50072943(CHEMBL3410310)
Affinity DataKi:  5.70E+3nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cells by Top Count analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
National University Of Singapore

Curated by ChEMBL
LigandPNGBDBM50072943(CHEMBL3410310)
Affinity DataKi: >2.00E+4nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-induced adenylyl cyclase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed