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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
7
hits in this display
Target
Kallikrein-7
(Homo sapiens (Human))
Sixera Pharma
US Patent
Ligand
BDBM113060
(US9695194, 1)
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Affinity Data
Ki: 48nM ΔG°: -43.5kJ/mole
pH: 7.2 T: 2°C
Assay Description:
Materials: Recombinant human KLK7, Substrate S-2586 (Chromogenics, cat. no. 820894) KLK7 activity was determined at 37° C. in 10 mM Na phosphate ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
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PC cid
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US Patent
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Target
Kallikrein-14
(Homo sapiens (Human))
Sixera Pharma
US Patent
Ligand
BDBM113060
(US9695194, 1)
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Affinity Data
Ki: 100nM ΔG°: -41.6kJ/mole
pH: 8.0 T: 2°C
Assay Description:
Materials: Recombinant human KLK14, Substrate S-2302 (Chromogenics, cat. no. 820340). KLK14 activity was determined at 37° C. in 0.1 mM Tris, pH ...
More data for this Ligand-Target Pair
Target Info
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KEGG
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antibodypedia
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US Patent
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Target
Kallikrein-5 [D153N]
(Homo sapiens (Human))
Sixera Pharma
US Patent
Ligand
BDBM113060
(US9695194, 1)
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Affinity Data
Ki: 200nM ΔG°: -39.8kJ/mole
pH: 8.0 T: 2°C
Assay Description:
Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...
More data for this Ligand-Target Pair
Target Info
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MMDB
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Ligand Info
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US Patent
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Target
Serine protease 1
(Homo sapiens (Human))
Sixera Pharma
US Patent
Ligand
BDBM113060
(US9695194, 1)
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Affinity Data
Ki: >1.00E+4nM ΔG°: >-29.7kJ/mole
pH: 7.2 T: 2°C
Assay Description:
Materials: Trypsin, 100 ug (Roche, sequence grade, Mw 23500), Substrate S-2288 (Chromogenics, cat. no. 820852). Trypsin activity was determined at 3...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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KEGG
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DrugBank
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Ligand Info
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PC sid
In Depth
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US Patent
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Target
Chymotrypsin-C
(Homo sapiens (Human))
Sixera Pharma
US Patent
Ligand
BDBM113060
(US9695194, 1)
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Affinity Data
Ki: >1.00E+4nM ΔG°: >-29.7kJ/mole
pH: 7.2 T: 2°C
Assay Description:
Materials: Chymotrypsin, bovine, 25 ug (Roche, sequence grade), Substrate S-2586 (Chromogenics, cat. no. 82 08 94). Chymotrypsin activity was determi...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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antibodypedia
GoogleScholar
Ligand Info
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PC cid
PC sid
In Depth
Details
US Patent
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Target
Prothrombin
(Homo sapiens (Human))
Sixera Pharma
US Patent
Ligand
BDBM113060
(US9695194, 1)
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Affinity Data
Ki: >1.00E+4nM ΔG°: >-29.7kJ/mole
pH: 8.3 T: 2°C
Assay Description:
Materials: Thrombin (Chromogenics, cat. no. 820712), Substrate S-2288 (Chromogenics, cat. no. 82 08 52). Thrombin activity was determined at 37° ...
More data for this Ligand-Target Pair
Target Info
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PC cid
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US Patent
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Target
Cathepsin G
(Homo sapiens (Human))
Sixera Pharma
US Patent
Ligand
BDBM113060
(US9695194, 1)
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Affinity Data
Ki: >1.00E+4nM ΔG°: >-29.7kJ/mole
pH: 7.2 T: 2°C
Assay Description:
Materials: Cathepsin G, 100 mU (VWR, Calbiochem, cat. no. 219373), Substrate Cathepsin G substrate (VWR, Calbiochem, cat. no. 219407). Cathepsin acti...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
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KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI