Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetImportin subunit alpha-1(Homo sapiens (Human))
Broad Institute

Curated by PubChem BioAssay

LigandBDBM62798(3-(4-ethoxy-3-methoxy-phenyl)-2-(4-fluorophenyl)-5...)Copy SMILESCopy InChI

Affinity DataEC50:  2.39E+5nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

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In DepthDetails PCBioAssay
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TargetHeat shock factor protein 1(Mus musculus)
Broad Institute

Curated by PubChem BioAssay

LigandBDBM62798(3-(4-ethoxy-3-methoxy-phenyl)-2-(4-fluorophenyl)-5...)Copy SMILESCopy InChI

Affinity DataEC50: >1.95E+5nMAssay Description:Keywords: Heat Shock Factor-1 (HSF-1), Stress Response, MG132, NIH3T3, Luminescence Assay Overview: Modified NIH3T3, transformed to express firefly...More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADGoogleScholar

Ligand InfoPurchasePC cidPC sidSimilars

In DepthDetails PCBioAssay
Copy BDB DOI