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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetKynurenine/alpha-aminoadipate aminotransferase, mitochondrial(Rattus norvegicus)
Tes Pharma

Curated by ChEMBL
LigandPNGBDBM50126148(CHEMBL3629572)
Affinity DataIC50:  7.10E+4nMAssay Description:Inhibition of rat liver KAT2 using [3H]-kynurenine incubated for 2 hrs by liquid scintillation spectrometry methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKynurenine/alpha-aminoadipate aminotransferase, mitochondrial(Rattus norvegicus)
Tes Pharma

Curated by ChEMBL
LigandPNGBDBM50126148(CHEMBL3629572)
Affinity DataIC50:  7.10E+4nMAssay Description:Inhibition of rat KAT-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed