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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
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kcal/mol
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Found
1
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Target
A disintegrin and metalloproteinase with thrombospondin motifs 5 [262-930,L692P]
(Homo sapiens (Human))
Wyeth Research
Ligand
BDBM24004
(5-ethyl-5'-(4-methoxyphenyl)-1,2-dihydro-3'H-spiro...)
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Affinity Data
IC50: 1.40E+3nM
pH: 7.5 T: 2°C
Assay Description:
ADAMTS-5 activity was determined using a fluorescence resonance energy transfer (FRET) assay using a QF peptide containing an aggrecanase cleavage si...
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