Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50049679(6-(4,5-Dihydro-1H-imidazol-2-yl)-2-ethyl-10,10-dio...)
Affinity DataKi:  4nMAssay Description:Ex vivo value for inhibition of MAO A of rats sacrificed 2 hr after po administrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50049679(6-(4,5-Dihydro-1H-imidazol-2-yl)-2-ethyl-10,10-dio...)
Affinity DataIC50:  10nMAssay Description:Inhibitory concentration against rat brain mitochondrial monoamine oxidase AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed