Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetType-1 angiotensin II receptor(RABBIT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043431(3-[5-(2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridi...)
Affinity DataIC50:  170nMAssay Description:In vitro antagonist activity against angiotensin II receptor type 1 in rabbit aorta using [125I]-Sar, Ile AII.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043431(3-[5-(2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridi...)
Affinity DataIC50:  1.60E+4nMAssay Description:In vitro antagonist activity against angiotensin II receptor type 2 in rat midbrain using [125I]-Sar,Ile AII.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed