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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Type-1 angiotensin II receptor
(RABBIT)
The M. S. University Of Baroda
Curated by
ChEMBL
Ligand
BDBM50043434
(2-Ethyl-5,7-dimethyl-4-{1-[phenyl-(1H-tetrazol-5-y...)
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Affinity Data
IC50: 1nM
Assay Description:
Binding affinity to angiotensin AT1 receptor in rabbit aortic rings
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Type-1 angiotensin II receptor
(RABBIT)
The M. S. University Of Baroda
Curated by
ChEMBL
Ligand
BDBM50043434
(2-Ethyl-5,7-dimethyl-4-{1-[phenyl-(1H-tetrazol-5-y...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 18nM
Assay Description:
In vitro antagonist activity against angiotensin II receptor type 1 in rabbit aorta using [125I]-Sar, Ile AII.
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Type-2 angiotensin II receptor
(RAT)
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50043434
(2-Ethyl-5,7-dimethyl-4-{1-[phenyl-(1H-tetrazol-5-y...)
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Copy InChI
Affinity Data
IC50: >3.00E+4nM
Assay Description:
In vitro antagonist activity against angiotensin II receptor type 2 in rat midbrain using [125I]-Sar,Ile AII.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI