Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetAdenosine receptor A3(Homo sapiens (Human))
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149118(5-Ethyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo...)
Affinity DataIC50:  6.20nMAssay Description:Displacement of specific [125I]-AB-MECA binding at human adenosine A3 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149118(5-Ethyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo...)
Affinity DataIC50:  27nMAssay Description:Displacement of specific [3H]-DPCPX binding at human adenosine A1 receptor expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149118(5-Ethyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo...)
Affinity DataIC50: <100nMAssay Description:Displacement of specific [3H]DPCPX binding at human adenosine A2B receptor expressed in HEK293 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Otsuka Pharmaceutical Factory

Curated by ChEMBL
LigandPNGBDBM50149118(5-Ethyl-2-phenyl-7H-pyrazolo[4,3-e][1,2,4]triazolo...)
Affinity DataIC50:  310nMAssay Description:Displacement of specific [3H]-CGS- 21680 binding at human adenosine A2A receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed