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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015746(1-Ethyl-7-fluoro-[1,2,4]triazolo[4,3-a]quinoxalin-...)
Affinity DataIC50:  170nMAssay Description:Evaluated for the binding affinity towards the Adenosine A2 receptor in corpora striata of rats using [3H]NECA as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50015746(1-Ethyl-7-fluoro-[1,2,4]triazolo[4,3-a]quinoxalin-...)
Affinity DataIC50:  580nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed