Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 5 hits in this display
BDBM50015749((1-Ethyl-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)-is...)
BDBM50015749((1-Ethyl-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)-is...)
BDBM50015749((1-Ethyl-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)-is...)
IC50: 660nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
BDBM50015749((1-Ethyl-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)-is...)
BDBM50015749((1-Ethyl-[1,2,4]triazolo[4,3-a]quinoxalin-4-yl)-is...)
IC50: 6.40E+3nMAssay Description:Evaluated for the binding affinity towards the Adenosine A2 receptor in corpora striata of rats using [3H]NECA as radioligand.More data for this Ligand-Target Pair