Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAdenosine receptor A1(Rattus norvegicus (rat))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50023487(Bicyclo[2.2.1]hept-2-yl-(1-ethyl-[1,2,4]triazolo[4...)
Affinity DataKi:  44nMAssay Description:Binding affinity towards adenosine A1 receptor using [3H]-N-cyclohexyladenosine in rat whole brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50023487(Bicyclo[2.2.1]hept-2-yl-(1-ethyl-[1,2,4]triazolo[4...)
Affinity DataKi:  6.10E+3nMAssay Description:Binding affinity against Adenosine-2 receptor with [3H]-NECA in rat striatal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed