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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAdenosine receptor A2a/A2b(Rattus norvegicus)
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50018577(5,7-Diethyl-2-phenyl-1,5-dihydro-imidazo[4,5-g]qui...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity against Adenosine A2 receptor in rat brain membrane, using [3H]-NECA as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of South Florida

Curated by ChEMBL
LigandPNGBDBM50018577(5,7-Diethyl-2-phenyl-1,5-dihydro-imidazo[4,5-g]qui...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity against Adenosine A1 receptor in rat brain membrane, using [3H]-N6-cyclohexyladenosine as the radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed