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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

LigandPNGBDBM50280879(12,13-diethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a...)
Affinity DataIC50:  200nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetcGMP-dependent protein kinase 1(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50280879(12,13-diethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a...)
Affinity DataIC50:  700nMAssay Description:In vitro for inhibitory activity against cGMP-dependent protein kinase from bovine lung (G-kinase)More data for this Ligand-Target Pair
In DepthDetails Article
TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
TBA

Curated by ChEMBL
LigandPNGBDBM50280879(12,13-diethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a...)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro for inhibitory activity against myosin light-chain kinase from chicken gizzard (M-kinase)More data for this Ligand-Target Pair
In DepthDetails Article
TargetcAMP-dependent protein kinase catalytic subunit alpha(Bos taurus (bovine))
TBA

Curated by ChEMBL
LigandPNGBDBM50280879(12,13-diethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro for inhibitory activity against cAMP-dependent protein kinase from bovine heart (A-kinase)More data for this Ligand-Target Pair
In DepthDetails Article