Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 31 hits in this display
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
Ki: 2.30nMAssay Description:Concentration that inhibits the binding of radioligand, [3H]-ICS 205930, to 5-hydroxytryptamine 3 receptor from rat cortexMore data for this Ligand-Target Pair
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
Ki: 4nMAssay Description:Tested for its binding affinity by measuring its ability to displace [3H]granisetron from 5-hydroxytryptamine 3 receptor in rat cortexMore data for this Ligand-Target Pair
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
BDBM50007872(3-Ethyl-2-oxo-2,3-dihydro-benzoimidazole-1-carboxy...)
EC50: 10nMAssay Description:Tested for its agonist potency against the 5-hydroxytryptamine 4 receptor located in the rat esophageal tunica muscularis mucosaeMore data for this Ligand-Target Pair