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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
D(2) dopamine receptor
(BOVINE)
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50017524
(7-Chloro-2-ethyl-10-(4-methyl-piperazin-1-yl)-2,4-...)
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Affinity Data
IC50: 67nM
Assay Description:
Inhibitory activity against dopamine receptor D2 in calf caudate tissue using [3H]spiperone
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Muscarinic acetylcholine receptor M1/M2/M3/M4/M5
(RAT)
Eli Lilly
Curated by
ChEMBL
Ligand
BDBM50017524
(7-Chloro-2-ethyl-10-(4-methyl-piperazin-1-yl)-2,4-...)
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Copy InChI
Affinity Data
IC50: 2.40E+3nM
Assay Description:
Inhibitory activity against muscarinic cholinergic receptors in male olac rat brain, using [3H]QNB as the radioligand
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI