Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063059(CHEMBL3398390)
Affinity DataIC50:  702nMAssay Description:Displacement of [3H]Ketanserin from human recombinant 5-HT2A receptor expressed in CHO-K1 cells after 15 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50063059(CHEMBL3398390)
Affinity DataIC50:  4.97E+3nMAssay Description:Inhibition of human recombinant 5-HT6 receptor expressed in HEK293 cells assessed as inhibition of 5-HT-induced increase in Ca2+ level pretreated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed