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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
7
hits in this display
Target
Coagulation factor X
(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50114452
(2-[3-(N,N-Dimethyl-carbamimidoyl)-naphthalen-2-yl]...)
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Affinity Data
IC50: 1.65E+3nM
Assay Description:
Inhibitory activity against coagulation factor Xa
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Plasminogen
(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50114452
(2-[3-(N,N-Dimethyl-carbamimidoyl)-naphthalen-2-yl]...)
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Affinity Data
IC50: >1.10E+4nM
Assay Description:
Inhibitory activity against tissue plasminogen activator
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Vitamin K-dependent protein C
(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50114452
(2-[3-(N,N-Dimethyl-carbamimidoyl)-naphthalen-2-yl]...)
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Affinity Data
IC50: >1.10E+4nM
Assay Description:
Inhibitory activity against activated protein C
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Plasminogen
(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50114452
(2-[3-(N,N-Dimethyl-carbamimidoyl)-naphthalen-2-yl]...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.10E+4nM
Assay Description:
Inhibitory activity against tissue plasminogen activator
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Prothrombin
(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50114452
(2-[3-(N,N-Dimethyl-carbamimidoyl)-naphthalen-2-yl]...)
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Copy InChI
Affinity Data
IC50: >1.10E+4nM
Assay Description:
Inhibitory activity against thrombin
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Kallikrein-1
(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50114452
(2-[3-(N,N-Dimethyl-carbamimidoyl)-naphthalen-2-yl]...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.10E+4nM
Assay Description:
Inhibitory activity against kallikrein
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine protease 1
(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50114452
(2-[3-(N,N-Dimethyl-carbamimidoyl)-naphthalen-2-yl]...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.10E+4nM
Assay Description:
Inhibitory activity against trypsin
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI