Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Homo sapiens (Human))
Bioland Laboratory (Guangzhou Regenerative Medicine And Health - Guangdong Laboratory)

Curated by ChEMBL
LigandPNGBDBM50066136(CHEMBL3400291)
Affinity DataIC50:  172nMAssay Description:Inhibition of PI3Kalpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
The University Of Michigan Medical School

Curated by ChEMBL
LigandPNGBDBM50066136(CHEMBL3400291)
Affinity DataIC50:  473nMAssay Description:Inhibition of MEK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
The University Of Michigan Medical School

Curated by ChEMBL
LigandPNGBDBM50066136(CHEMBL3400291)
Affinity DataIC50:  473nMAssay Description:Inhibition of MEK1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
The University Of Michigan Medical School

Curated by ChEMBL
LigandPNGBDBM50066136(CHEMBL3400291)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of PKC-alpha (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
The University Of Michigan Medical School

Curated by ChEMBL
LigandPNGBDBM50066136(CHEMBL3400291)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of AurB (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
The University Of Michigan Medical School

Curated by ChEMBL
LigandPNGBDBM50066136(CHEMBL3400291)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed