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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
B2 bradykinin receptor
(Homo sapiens (Human))
Fujisawa Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50142955
(4-{(E)-2-[({[2,4-Dichloro-3-(4-imidazol-1-yl-2-met...)
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Affinity Data
IC50: 0.350nM
Assay Description:
In vitro inhibitory activity towards human bradykinin receptor B2 expressed in CHO cells using [3H]BK (1.0 nM) as a radioligand
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
B2 bradykinin receptor
(Homo sapiens (Human))
Fujisawa Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50142955
(4-{(E)-2-[({[2,4-Dichloro-3-(4-imidazol-1-yl-2-met...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 4.30nM
Assay Description:
In vitro inhibitory activity towards bradykinin receptor B2 using [3H]BK (0.06 nM) as a radioligand in guinea pig ileum membrane preparation
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI