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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
C-X-C chemokine receptor type 2
(Homo sapiens (Human))
Galderma Research & Development
US Patent
Ligand
BDBM236781
(US9388149, 12 | US9580412, Example 12)
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Affinity Data
IC50: 83nM
T: 2°C
Assay Description:
PathHunter HEK293-CXCR2 or U2OS hCXCR1 β-arrestin cells (DiscoveRx Corporation) were seeded overnight at 10 000 cells/well (384-well...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
C-X-C chemokine receptor type 2
(Homo sapiens (Human))
Galderma Research & Development
US Patent
Ligand
BDBM236781
(US9388149, 12 | US9580412, Example 12)
Copy SMILES
Copy InChI
Affinity Data
IC50: 83nM
Assay Description:
The in vitro affinity of the compounds of the present invention for the CXCR1 and CXCR2 receptors was determined on a functional test of the β-a...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
C-X-C chemokine receptor type 1
(Homo sapiens (Human))
Galderma Research & Development
US Patent
Ligand
BDBM236781
(US9388149, 12 | US9580412, Example 12)
Copy SMILES
Copy InChI
Affinity Data
IC50: 483nM
Assay Description:
The in vitro affinity of the compounds of the present invention for the CXCR1 and CXCR2 receptors was determined on a functional test of the β-a...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
C-X-C chemokine receptor type 1
(Homo sapiens (Human))
Galderma Research & Development
US Patent
Ligand
BDBM236781
(US9388149, 12 | US9580412, Example 12)
Copy SMILES
Copy InChI
Affinity Data
IC50: 483nM
T: 2°C
Assay Description:
PathHunter HEK293-CXCR2 or U2OS hCXCR1 β-arrestin cells (DiscoveRx Corporation) were seeded overnight at 10 000 cells/well (384-well...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI