Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50242675(CHEMBL453043 | N,N-Dimethyl-5-((7-phenylheptanamid...)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of FAAH mediated [14C]anadamide hydrolysis in rat brain after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol lipase-alpha(Homo sapiens (Human))
Sapienza University Of Rome

Curated by ChEMBL
LigandPNGBDBM50242675(CHEMBL453043 | N,N-Dimethyl-5-((7-phenylheptanamid...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human recombinant DAGLalpha mediated sn-1-[14C]oleoyl-2-arachidonoyl-glycerol hydrolysis to 2-AG overexpressed in COS cells after 20 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed