Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL

LigandBDBM50201281(CHEMBL234253 | dimethyl-{3-[(2-p-tolyl-ethylamino)...)Copy SMILESCopy InChI

Affinity DataKi:  18nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL

LigandBDBM50201281(CHEMBL234253 | dimethyl-{3-[(2-p-tolyl-ethylamino)...)Copy SMILESCopy InChI

Affinity DataKi:  48nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M2 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Mitsubishi Pharma

Curated by ChEMBL

LigandBDBM50201281(CHEMBL234253 | dimethyl-{3-[(2-p-tolyl-ethylamino)...)Copy SMILESCopy InChI

Affinity DataKi:  220nMAssay Description:Displacement of 1-[N-methyl- 3H]scopolamine from human muscarinic M1 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair

Target InfoReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI