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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
31
hits in this display
Target
Tyrosine-protein kinase receptor TYRO3
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 2nM
Assay Description:
Inhibition of Sky (unknown origin) by ELISA kinase assay in presence of 60 uM ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
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Target
Mitogen-activated protein kinase kinase kinase kinase 4
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 120nM
Assay Description:
Inhibition of MAP4K4 (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
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Target
P-selectin
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 400nM
Assay Description:
Inhibition of P-selectin aggregation in platelet surface (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
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KEGG
UniProtKB/SwissProt
B.MOAD
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Target
Tyrosine-protein kinase Lck
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 610nM
Assay Description:
Inhibition of LCK (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
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Target
Dual specificity protein kinase CLK1
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 3.45E+3nM
Assay Description:
Inhibition of CLK1 (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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Target
Tyrosine-protein kinase ABL1
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 7.61E+3nM
Assay Description:
Inhibition of ABL (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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UniProtKB/SwissProt
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Target
Myosin light chain kinase 2, skeletal/cardiac muscle
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 8.27E+3nM
Assay Description:
Inhibition of MYLK2 (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
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Target
Mitogen-activated protein kinase kinase kinase 9
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 1.22E+4nM
Assay Description:
Inhibition of MAP3K9 (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
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Target
Calcium/calmodulin-dependent protein kinase type 1
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 1.97E+4nM
Assay Description:
Inhibition of CAMK1 (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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KEGG
UniProtKB/SwissProt
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CHEMBL
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Target
Tyrosine-protein kinase JAK3
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of JAK3 (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
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KEGG
UniProtKB/SwissProt
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PubMed
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Target
Insulin receptor
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of INSR (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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KEGG
UniProtKB/SwissProt
B.MOAD
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Target
Inhibitor of nuclear factor kappa-B kinase subunit epsilon
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of IKKi (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
Reactome pathway
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CHEMBL
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Target
Inhibitor of nuclear factor kappa-B kinase subunit beta
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of IKK-beta (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
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Target
Glycogen synthase kinase-3 beta
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of GSK3-beta (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
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Article
PubMed
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Target
Fibroblast growth factor receptor 1
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of FGFR1 (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
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Article
PubMed
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Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of EGFR (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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Article
PubMed
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Target
Ephrin type-A receptor 2
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of ECK (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Serine/threonine-protein kinase Chk2
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of CHK2 (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Tyrosine-protein kinase BTK
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of BTK (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Aurora kinase A
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of Aurora-A (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
RAC-alpha serine/threonine-protein kinase
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Copy InChI
Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of AKT1 (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mitogen-activated protein kinase 1
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
Copy SMILES
Copy InChI
Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of MAPK1/ERK2 (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
MAP kinase-activated protein kinase 2
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of MAPKAP-K2 (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase MARK1
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
Copy SMILES
Copy InChI
Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of MARK1 (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 26
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
Copy SMILES
Copy InChI
Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of MASK (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase 3
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
Copy SMILES
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Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of MST2 (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase Nek2
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of NEK2 (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase Chk1
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
Copy SMILES
Copy InChI
Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of CHK1 (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Serine/threonine-protein kinase PAK 4
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of PAK4 (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Cyclin-dependent kinase 6/G1/S-specific cyclin-D3
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of CDK6/cyclin D3 (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
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Article
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Target
Cyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2
(Homo sapiens (Human))
Pfizer
Curated by
ChEMBL
Ligand
BDBM50425864
(CHEMBL2312649)
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Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of CDK2/cyclin A (unknown origin) in presence of ATP
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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