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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Muscarinic acetylcholine receptor M2
(RAT)
Dr. Karl Thomae
Curated by
ChEMBL
Ligand
BDBM50018297
(11-[2-(2-Dimethylaminomethyl-piperidin-1-yl)-acety...)
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Affinity Data
IC50: 140nM
Assay Description:
Binding affinity to the rat cardiac muscarinic acetylcholine receptor M2 using 0.3 nM [3H]-N-methylscopolamine as radioligand
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M2
(RAT)
Dr. Karl Thomae
Curated by
ChEMBL
Ligand
BDBM50018297
(11-[2-(2-Dimethylaminomethyl-piperidin-1-yl)-acety...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 140nM
Assay Description:
Inhibition of muscarinic (M2) receptor isolated from rat atria
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M3
(RAT)
College Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50018297
(11-[2-(2-Dimethylaminomethyl-piperidin-1-yl)-acety...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.00E+3nM
Assay Description:
Inhibition of rat submandibular muscarinic (M3) receptor isolated from tissue homogenates
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Muscarinic acetylcholine receptor M3
(RAT)
College Of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50018297
(11-[2-(2-Dimethylaminomethyl-piperidin-1-yl)-acety...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.00E+3nM
Assay Description:
Binding affinity for glandular muscarinic acetylcholine receptor M3 in rat assayed using 0.3 nM [3H]-N-methylscopolamine as radioligand
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI