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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetAlpha-2A/Alpha-2B/Alpha-2C adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50225334(CHEMBL281064)
Affinity DataKi:  25nMAssay Description:Binding affinity towards alpha 2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50225334(CHEMBL281064)
Affinity DataKi:  25nMAssay Description:Binding affinity towards alpha-2 adrenergic receptor in rat using [3H]rauwolscine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50225334(CHEMBL281064)
Affinity DataKi:  6.90E+3nMAssay Description:Binding affinity against alpha-1 adrenergic receptor in rat using [3H]prazosin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50225334(CHEMBL281064)
Affinity DataKi:  6.90E+3nMAssay Description:Binding affinity towards alpha 1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed