Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetC-X-C chemokine receptor type 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL

LigandBDBM50193981(6-chloro-3-[((cyanoimino){[2-(trifluoromethyl)phen...)Copy SMILESCopy InChI

Affinity DataIC50:  12nMAssay Description:Displacement of [125I]IL8 from CXCR2 expressed in CHO cellsMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL

LigandBDBM50193981(6-chloro-3-[((cyanoimino){[2-(trifluoromethyl)phen...)Copy SMILESCopy InChI

Affinity DataIC50:  411nMAssay Description:Displacement of [125I]IL8 from CXCR1 expressed in CHO cellsMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI