Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343728(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343728(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-UR-MK114 from Y1R in human SK-N-MC cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343728(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi: >400nMAssay Description:Displacement of Dy-635-pNPY from human Y5R expressed in CHO cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343728(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi: >500nMAssay Description:Displacement of Cy5-[K4]-hpp from human Y4R expressed in CHO cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343728(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKi: >500nMAssay Description:Displacement of Dy-635-pNPY from human Y2R expressed in CHO cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 4(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343728(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of Cy5-[K4]-hpp from human Y4R expressed in CHO cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343728(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of Dy-635-pNPY from human Y5R expressed in CHO cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343728(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of Dy-635-pNPY from human Y2R expressed in CHO cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Universit£T Regensburg

Curated by ChEMBL
LigandPNGBDBM50343728(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKd:  5nMAssay Description:Binding affinity at Y1R in human MCF-7 cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed