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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188533(CHEMBL411335 | H-Tyr-Pro-Phe-Phe-NH-(CH2)5-(C=O)-D...)
Affinity DataKi:  245nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188533(CHEMBL411335 | H-Tyr-Pro-Phe-Phe-NH-(CH2)5-(C=O)-D...)
Affinity DataKi:  5.94E+3nMAssay Description:Displacement of [3H]deltorphin C from rat delta opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188533(CHEMBL411335 | H-Tyr-Pro-Phe-Phe-NH-(CH2)5-(C=O)-D...)
Affinity DataIC50:  253nMAssay Description:Functional bioactivity against mu opioid receptor in guinea-pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50188533(CHEMBL411335 | H-Tyr-Pro-Phe-Phe-NH-(CH2)5-(C=O)-D...)
Affinity DataIC50:  300nMAssay Description:Functional bioactivity against delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed