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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Mu-type opioid receptor
(Rattus norvegicus (rat))
Universidad De Santiago De Compostela
Curated by
ChEMBL
Ligand
BDBM50188533
(CHEMBL411335 | H-Tyr-Pro-Phe-Phe-NH-(CH2)5-(C=O)-D...)
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Affinity Data
Ki: 245nM
Assay Description:
Displacement of [3H]DAMGO from rat mu opioid receptor in brain P2 synaptosomes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Delta-type opioid receptor
(Rattus norvegicus (rat))
Universidad De Santiago De Compostela
Curated by
ChEMBL
Ligand
BDBM50188533
(CHEMBL411335 | H-Tyr-Pro-Phe-Phe-NH-(CH2)5-(C=O)-D...)
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Copy InChI
Affinity Data
Ki: 5.94E+3nM
Assay Description:
Displacement of [3H]deltorphin C from rat delta opioid receptor in brain P2 synaptosomes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mu-type opioid receptor
(GUINEA PIG)
Universidad De Santiago De Compostela
Curated by
ChEMBL
Ligand
BDBM50188533
(CHEMBL411335 | H-Tyr-Pro-Phe-Phe-NH-(CH2)5-(C=O)-D...)
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Affinity Data
IC50: 253nM
Assay Description:
Functional bioactivity against mu opioid receptor in guinea-pig ileum
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Delta-type opioid receptor
(MOUSE)
Universidad De Santiago De Compostela
Curated by
ChEMBL
Ligand
BDBM50188533
(CHEMBL411335 | H-Tyr-Pro-Phe-Phe-NH-(CH2)5-(C=O)-D...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 300nM
Assay Description:
Functional bioactivity against delta opioid receptor in mouse vas deferens
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI