Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
University Of Pavia

Curated by ChEMBL

LigandBDBM50357428(CHEMBL1917701)Copy SMILESCopy InChI

Affinity DataKi:  92nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetMu-type opioid receptor(GUINEA PIG)
University Of Pavia

Curated by ChEMBL

LigandBDBM50357428(CHEMBL1917701)Copy SMILESCopy InChI

Affinity DataKi:  119nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
B.MOADGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Pavia

Curated by ChEMBL

LigandBDBM50357428(CHEMBL1917701)Copy SMILESCopy InChI

Affinity DataKi:  438nMAssay Description:Displacement of [3H]-U69593 from kappa opioid receptor in guinea pig brain membrane after 150 mins by liquid scintillation countingMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
B.MOADGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI