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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

LigandPNGBDBM50013849(14-[4-azido(methyl)anilino]-4-cyclopropylmethyl-12...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50013849(14-[4-azido(methyl)anilino]-4-cyclopropylmethyl-12...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50013849(14-[4-azido(methyl)anilino]-4-cyclopropylmethyl-12...)
Affinity DataKi:  0.700nMAssay Description:Opioid receptor delta 1 apparent binding constant from rat brain membranes using [3H]DADLE binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50013849(14-[4-azido(methyl)anilino]-4-cyclopropylmethyl-12...)
Affinity DataKi:  0.700nMAssay Description:Opioid receptor kappa 1 apparent binding constant from guinea pig cerebellum using [3H]diprenorphine binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed