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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM225266(2-((5-Chloro-2-hydroxyphenyl)(methyl)amino)-N-(3-(...)
Affinity DataIC50:  9.50E+3nMpH: 7.5 T: 2°CAssay Description:The LSD1 screening biochemical assay was performed by Shanghai ChemPartner Co. Ltd and the detailed protocol was shown as followed. The AlphaLISA ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM225266(2-((5-Chloro-2-hydroxyphenyl)(methyl)amino)-N-(3-(...)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of human LSD1 (158 to end residues) expressed in Escherichia coli preincubated for 15 mins followed by H3K4me2 peptide addition and measur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM225266(2-((5-Chloro-2-hydroxyphenyl)(methyl)amino)-N-(3-(...)
Affinity DataIC50:  6.57E+4nMAssay Description:The MAO-A and MAO-B is purchased from Active Motif (Cat#31502, Cat#31503). Biochemical Kit is purchased from Promega (MAO-Glo Assay, V1402). The inhi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
China Pharmaceutical University

LigandPNGBDBM225266(2-((5-Chloro-2-hydroxyphenyl)(methyl)amino)-N-(3-(...)
Affinity DataIC50:  1.87E+5nMAssay Description:The MAO-A and MAO-B is purchased from Active Motif (Cat#31502, Cat#31503). Biochemical Kit is purchased from Promega (MAO-Glo Assay, V1402). The inhi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed