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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Lysine-specific histone demethylase 1A
(Homo sapiens (Human))
China Pharmaceutical University
Ligand
BDBM225266
(2-((5-Chloro-2-hydroxyphenyl)(methyl)amino)-N-(3-(...)
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Affinity Data
IC50: 9.50E+3nM
pH: 7.5 T: 2°C
Assay Description:
The LSD1 screening biochemical assay was performed by Shanghai ChemPartner Co. Ltd and the detailed protocol was shown as followed. The AlphaLISA ass...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Lysine-specific histone demethylase 1A
(Homo sapiens (Human))
China Pharmaceutical University
Ligand
BDBM225266
(2-((5-Chloro-2-hydroxyphenyl)(methyl)amino)-N-(3-(...)
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Copy InChI
Affinity Data
IC50: 9.50E+3nM
Assay Description:
Inhibition of human LSD1 (158 to end residues) expressed in Escherichia coli preincubated for 15 mins followed by H3K4me2 peptide addition and measur...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Amine oxidase [flavin-containing] B
(Homo sapiens (Human))
China Pharmaceutical University
Ligand
BDBM225266
(2-((5-Chloro-2-hydroxyphenyl)(methyl)amino)-N-(3-(...)
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Affinity Data
IC50: 6.57E+4nM
Assay Description:
The MAO-A and MAO-B is purchased from Active Motif (Cat#31502, Cat#31503). Biochemical Kit is purchased from Promega (MAO-Glo Assay, V1402). The inhi...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Amine oxidase [flavin-containing] A
(Homo sapiens (Human))
China Pharmaceutical University
Ligand
BDBM225266
(2-((5-Chloro-2-hydroxyphenyl)(methyl)amino)-N-(3-(...)
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Copy InChI
Affinity Data
IC50: 1.87E+5nM
Assay Description:
The MAO-A and MAO-B is purchased from Active Motif (Cat#31502, Cat#31503). Biochemical Kit is purchased from Promega (MAO-Glo Assay, V1402). The inhi...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI