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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human))
Abbott Laboratories
Curated by
ChEMBL
Ligand
BDBM50188755
(1-methyl-1-((5-(6-((4-methylpiperazin-1-yl)methyl)...)
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Affinity Data
IC50: 122nM
Assay Description:
Inhibition of KDR at 1 mM ATP by HTRF assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Vascular endothelial growth factor receptor 1
(Homo sapiens (Human))
Abbott Laboratories
Curated by
ChEMBL
Ligand
BDBM50188755
(1-methyl-1-((5-(6-((4-methylpiperazin-1-yl)methyl)...)
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Copy InChI
Affinity Data
IC50: 4.95E+3nM
Assay Description:
Inhibition of FLT1 at 1mM ATP by HTRF assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mast/stem cell growth factor receptor Kit
(Homo sapiens (Human))
Abbott Laboratories
Curated by
ChEMBL
Ligand
BDBM50188755
(1-methyl-1-((5-(6-((4-methylpiperazin-1-yl)methyl)...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 5.71E+3nM
Assay Description:
Inhibition of cKit at 1 mM ATP by HTRF assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI