Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50066173((S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(b...)
Affinity DataKi:  2.20nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Novartis Institute For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50066173((S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(b...)
Affinity DataIC50:  17nMAssay Description:Tachykinin receptor 1 agonistic activity as inhibition of contractions evoked by 4 nM [Sar9,Met(O2)11]-SP in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed