Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetPolyunsaturated fatty acid 5-lipoxygenase(Rattus norvegicus)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50003445(3-(Hydroxy-methyl-amino)-thioacrylic acid S-naphth...)
Affinity DataIC50:  240nMAssay Description:inhibitory activity against 5-lipoxygenase in rat basophilic leukemia cell line.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed