Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50314464((S)-N-((S)-1-cyclohexyl-2-((S)-2-(4-methylbenzo[d]...)
Affinity DataKi:  9.40E+5nMAssay Description:Antagonist activity at XIAP BIR3 domain by fluorescence polarization assay ... On Thursday, November 10, 2011 9:19 AM from cohen.fred@gene.com: Unfor...Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 7(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50314464((S)-N-((S)-1-cyclohexyl-2-((S)-2-(4-methylbenzo[d]...)
Affinity DataKi:  2.70E+6nMAssay Description:Antagonist activity at ML-IAP MLXBIR3SG domain by fluorescence polarization assay ... On Thursday, November 10, 2011 9:19 AM from cohen.fred@gene.com...Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed