Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM139080(US8883771, 26)
Affinity DataIC50: <1.00E+3nMpH: 7.5Assay Description:Binding affinities of the present compounds to XIAP linker-BIR2-BIR3 (residues 120-356), cIAP1-BIR3 (residues 253-363), and cIAP-2 BIR3 (residues 238...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBaculoviral IAP repeat-containing protein 3(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM139080(US8883771, 26)
Affinity DataIC50: <1.00E+3nMpH: 7.5Assay Description:Binding affinities of the present compounds to XIAP linker-BIR2-BIR3 (residues 120-356), cIAP1-BIR3 (residues 253-363), and cIAP-2 BIR3 (residues 238...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM139080(US8883771, 26)
Affinity DataIC50: <1.00E+3nMpH: 7.5Assay Description:Binding affinities of the present compounds to XIAP linker-BIR2-BIR3 (residues 120-356), cIAP1-BIR3 (residues 253-363), and cIAP-2 BIR3 (residues 238...More data for this Ligand-Target Pair
In DepthDetails US Patent