Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 8 hits in this display
BDBM50273699((5S,8S,10aR)-N-Benzhydryl-5-((S)-2-(methyl-amino)p...)
BDBM50273699((5S,8S,10aR)-N-Benzhydryl-5-((S)-2-(methyl-amino)p...)
Ki: 1.5nMAssay Description:Displacement of fluorescently tagged SM5F from human cIAP-1 BIR3 expressed in Escherichia coli BL21 cells by fluorescence polarization assayMore data for this Ligand-Target Pair
BDBM50273699((5S,8S,10aR)-N-Benzhydryl-5-((S)-2-(methyl-amino)p...)
Ki: 4.20nMAssay Description:Displacement of fluorescently tagged SM5F from human cIAP-2 BIR3 expressed in Escherichia coli BL21 cells by fluorescence polarization assayMore data for this Ligand-Target Pair
BDBM50273699((5S,8S,10aR)-N-Benzhydryl-5-((S)-2-(methyl-amino)p...)
BDBM50273699((5S,8S,10aR)-N-Benzhydryl-5-((S)-2-(methyl-amino)p...)
BDBM50273699((5S,8S,10aR)-N-Benzhydryl-5-((S)-2-(methyl-amino)p...)
IC50: 9nMAssay Description:Displacement of fluorescent SM5F peptide from His-tagged human cIAP1 BIR3 domain expressed in Escherichia coli BL21(DE3) cells by fluorescence polari...More data for this Ligand-Target Pair
BDBM50273699((5S,8S,10aR)-N-Benzhydryl-5-((S)-2-(methyl-amino)p...)
IC50: 26.3nMAssay Description:Displacement of fluorescent SM5F peptide from His-tagged human cIAP2 BIR3 domain expressed in Escherichia coli BL21(DE3) cells by fluorescence polari...More data for this Ligand-Target Pair
BDBM50273699((5S,8S,10aR)-N-Benzhydryl-5-((S)-2-(methyl-amino)p...)
IC50: 370nMAssay Description:Displacement of fluorescent SM5F peptide from His-tagged human XIAP BIR3 domain expressed in Escherichia coli BL21(DE3) cells by fluorescence polariz...More data for this Ligand-Target Pair