Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 15 hits in this display   

TargetNorepinephrine transporter(RAT)
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
Affinity DataKi:  0.260nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Toronto

Curated by PDSP Ki Database
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
Affinity DataKi:  0.410nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
Affinity DataKi:  0.480nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
Affinity DataKi:  0.990nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Toronto

Curated by PDSP Ki Database
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
In DepthDetails PubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Toronto

Curated by PDSP Ki Database
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
Affinity DataKi:  5.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNorepinephrine transporter(RAT)
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
Affinity DataKi:  8.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
Affinity DataKi:  11.9nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Toronto

Curated by PDSP Ki Database
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
Affinity DataKi:  290nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
Affinity DataKi:  740nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
University Of Toronto

Curated by PDSP Ki Database
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
Affinity DataKi:  890nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Lundbeck Ais

Curated by PDSP Ki Database
LigandPNGBDBM81946(CAS_96850-13-4 | LU 19,005 | LU 19-005)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed