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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50388014(CHEMBL2058420)
Affinity DataKi:  1.22E+3nMAssay Description:Displacement of [3H]GR65630 from human recombinant 5HT3 receptor expressed in HEKT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50388014(CHEMBL2058420)
Affinity DataIC50:  52nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate preincubated with compound for 15 mins measured after 20 mins by fluorometric ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50388014(CHEMBL2058420)
Affinity DataIC50:  3.12E+3nMAssay Description:Inhibition of human recombinant MAO-B using kynuramine as substrate preincubated with compound for 15 mins measured after 20 mins by fluorometric ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed