Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetA disintegrin and metalloproteinase with thrombospondin motifs 5 [262-930,L692P](Homo sapiens (Human))
Wyeth Research

LigandBDBM24017(1-methyl-5'-(4-methylphenyl)-1,2-dihydro-3'H-spiro...)Copy SMILESCopy InChI

Affinity DataIC50:  4.60E+3nMAssay Description:ADAMTS-5 activity was determined using a fluorescence resonance energy transfer (FRET) assay using a QF peptide containing an aggrecanase cleavage si...More data for this Ligand-Target Pair

Target InfoPDBMMDB
UniProtKB/SwissProt
B.MOADDrugBankGoogleScholar

Ligand InfoPurchasePC cidPC sidSimilars

In DepthDetails ArticlePubMed
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