Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070195((6aR,9R,10aR)-7-Methyl-4,6,6a,7,8,9,10,10a-octahyd...)
Affinity DataIC50:  220nMAssay Description:Displacement of [3H]-spiroperidol from D2 receptor in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070195((6aR,9R,10aR)-7-Methyl-4,6,6a,7,8,9,10,10a-octahyd...)
Affinity DataIC50:  350nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor in rat frontal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50070195((6aR,9R,10aR)-7-Methyl-4,6,6a,7,8,9,10,10a-octahyd...)
Affinity DataIC50:  510nMAssay Description:Displacement of [3H]yohimbine from Alpha-2 adrenergic receptor in rat frontal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerotonin 2 (5-HT2) receptor(RAT)
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070195((6aR,9R,10aR)-7-Methyl-4,6,6a,7,8,9,10,10a-octahyd...)
Affinity DataIC50:  520nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor in rat pre frontal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070195((6aR,9R,10aR)-7-Methyl-4,6,6a,7,8,9,10,10a-octahyd...)
Affinity DataIC50:  570nMAssay Description:Displacement of [3H]-SCH-23,390 from D1 receptor in rat striatumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Pharmacia & Upjohn

Curated by ChEMBL
LigandPNGBDBM50070195((6aR,9R,10aR)-7-Methyl-4,6,6a,7,8,9,10,10a-octahyd...)
Affinity DataIC50:  690nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed