Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 12 hits in this display   

TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50431028(CHEMBL2338333)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of recombinant KDR (unknown origin) by FRET-based Z'-LYTE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50431028(CHEMBL2338333)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of recombinant AKT2 (unknown origin) by FRET-based Z'-LYTE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50431028(CHEMBL2338333)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of recombinant AMPK A1/B1/G1 (unknown origin) by FRET-based Z'-LYTE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50431028(CHEMBL2338333)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of recombinant AKT1 (unknown origin) by FRET-based Z'-LYTE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Nek1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50431028(CHEMBL2338333)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of recombinant NEK1 (unknown origin) by FRET-based Z'-LYTE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50431028(CHEMBL2338333)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of recombinant IKBKB (unknown origin) by FRET-based Z'-LYTE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50431028(CHEMBL2338333)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of recombinant RPS6K1 (unknown origin) by FRET-based Z'-LYTE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50431028(CHEMBL2338333)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of recombinant RAF1 (unknown origin) by cascade reaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50431028(CHEMBL2338333)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of recombinant MEK1 (unknown origin) by cascade reaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50431028(CHEMBL2338333)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of recombinant MAPKAPK2 (unknown origin) by FRET-based Z'-LYTE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50431028(CHEMBL2338333)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of recombinant ERK2 (unknown origin) by FRET-based Z'-LYTE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50431028(CHEMBL2338333)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant MAPK14 (unknown origin) by FRET-based Z'-LYTE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed